| [1] | Asif, M., 2012. Study of clinically used and recently developed antimycobacterial agents. Orient Pharm Exp Med, 12: pp. 15-34. |
| |
| [2] | World Health Organization. Strategic framework to decrease the burden of TB/HIV documents WHO/CDS/TB. 2002; 296, WHO/HIVAIDS/2002, 2. Geneva, Switzerland: World Health Organization. |
| |
| [3] | World Health Organisation, Tuberculosis, Fact Sheet No. 104, 2007. http:// www.who.int/mediacentre/factsheets/who104/en/index.html/. |
| |
| [4] | WHO report 2008: The Stop TB Strategy, case reports, treatment outcomes and estimates of TB burden. http://www.who.int/tb/publications/global_report/2008/annex_3/en/index.html. |
| |
| [5] | Asif, M., Siddiqui, A.A., Husain, A., 2012. Quinolone derivatives as antitubercular drugs. Med Chem Res, 22(3): 1029-1042. |
| |
| [6] | Kamal, A., Azeeza, S., Malik, M.S., Shaik, A.A., and Rao, M.V. 2008. Efforts Towards the Development of New Antitubercular Agents: Potential for Thiolactomycin Based Compounds. J Pharm Pharmaceut Sci, 11 (2): 56s-80s. |
| |
| [7] | Nahid, P., Pai, M., and Hopewell, P.C. Advances in the diagnosis and treatment of tuberculosis. Proc Am Thorac Soc 2006; 3: 103-10. |
| |
| [8] | Nguyen, L., and Thompson, C.J., 2006. Foundations of antibiotic resistance in bacterial physiology: the mycobacterial paradigm. Trends Microbiol, 14: 304-12. |
| |
| [9] | WHO, 2005. Global tuberculosis control-surveillance, planning, financing (Geneva: World Health Organization). |
| |
| [10] | World Health Organization (WHO). Treatment of tuberculosis: guidelines for national programmes. 3rd edition. 2003. Geneva. |
| |
| [11] | Tripathi, R.P., Tewari, N., Dwivedi, N., and Tiwari, V.K., 2005. Fighting tuberculosis: An old disease with new challenges. Med Res Rev., 25: 93-131. |
| |
| [12] | Bastian, I., and Colebunders, R., 1999. Treatment and prevention of multidrug-resistant tuberculosis. Drugs, 58(4), 633-661. |
| |
| [13] | Ahmad, Z., Sharma, S., Khuller, GK., Singh, P., Faujdar, J., and Katoch, VM. 2006. Antimycobacterial activity of econazole against multidrug-resistant strains of Mycobacterium tuberculosis. Inter J Antimicrob Agents, 28(6): pp. 543-544. |
| |
| [14] | Aldrich, C. C., Bosshoff, H. I., and Remmel R. P., 2010. Antitubercular agents, In: Burger's Medicinal Chemistry, Drug Discovery and Development, vol. 7 Antiinfectives, Abraham, Understanding Tuberculosi-D. J. & Rotella, D. P. (Eds.), 7th ed., pp.713-812, Wiley, New York. |
| |
| [15] | Management of MDR-TB. A field guide A companion document to Guidelines for the programmatic management of drug-resistant tuberculosis. WHO/HTM/TB/2008.402, WHO Library Cataloguing-in-Publication Data: World Health Organization, 2009. |
| |
| [16] | Center for Disease Control. "Emergence of Mycobacterium tuberculosis with Extensive Resistance to Second-Line Drugs—Worldwide, 2000-2004". 2006, 55: 301-305. |
| |
| [17] | Grosset, J. H., 1992. Treatment of tuberculosis in HIV infection. Tuber Lung Dis, 73: 378-383. |
| |
| [18] | Centers for Disease Control and Prevention. 1982. Adverse drug reactions among children treated for tuberculosis. M.M.W.R. Morb. Mortal. Wkly. Rep., 29: 589-591. |
| |
| [19] | Cole, ST., and Alzari, P. M. 2007. Towards new tuberculosis drugs. Biochemical Society Transactions, 35(5): pp. 1321-1324. |
| |
| [20] | Glickman, S. W., Rasiel, E. B., Hamilton, C. D., Kubataev, A., and Schulman, K. A., 2006. Medicine. A portfolio model of drug development for tuberculosis. Science, 311, 1246-1247. |
| |
| [21] | Stahlmann R, Lode H. Toxicity of quinolones. Drugs, 1999, 58(Suppl. 2):37-42. |
| |
| [22] | Rieder, H.L., Arnadottir T., Trebucq A, and Enarson, D.A., 2001. Tuberculosis treatment: dangerous regimens? Inter J Tuberculosis & Lung Diseases. 5: pp. 1-3. |
| |
| [23] | Russell, D. G., 2001. Mycobacterium tuberculosis: here today, and here tomorrow. Nat Rev Mol Cell Biol, 2: 569-577. |
| |
| [24] | Smith, C. V., Sharma, V., and Sacchettini, J. C., 2004. TB drug discovery: Addressing issues of persistence and resistance. Tuberculosis, 84, 45-55. |
| |
| [25] | O'Brien, R. J., and Nunn, P. P. The need for new drugs against tuberculosis. Obstacles, opportunities, and next steps. Am J Respir Crit Care Med, 2001, 163, 1055-1058. |
| |
| [26] | Paramasivan, C. N., Sulochana, S., Kubendiran, G., Venkatesan, P., and Mitchison, D. A. 2005. Bactericidal action of gatifloxacin, rifampin, and isoniazid on logarithmic- and stationary-phase cultures of Mycobacterium tuberculosis. Antimicrob Agents Chemother, 49: 627-631. |
| |
| [27] | Somoskovi, A., Parsons, L. M., and Salfinger, M., 2001. The molecular basis of resistance to Isoniazid, Rifampin, and Pyrazinamide in Mycobacterium tuberculosis. Respir. Res., 2: 164-168. |
| |
| [28] | Farr, B.F. Rifamycins. In, Mandell, Douglas and Bennett's Principles and Practice of Infectious Diseases, 5th ed. (Mandell, G.L., Bennett, J.E., and Dolin, R., eds.) Churchill Livingstone, Philadelphia, 2000, pp. 348-361. |
| |
| [29] | Temple, M.E., Nahata, M.C. Rifapentine: its role in the treatment of tuberculosis. Annals of Pharmacotherapy, 1999, 33(11):1202-1210. |
| |
| [30] | Zhang, Y., 2004. Persistent and dormant tubercle bacilli and latent tuberculosis. Frontiers Bioscience, 1(9): pp. 1136-1156. |
| |
| [31] | Baciewicz, A.M., Self, T.H., and Bekemeyer, W.B., 1987. Update on rifampin drug interactions. Arch. Intern. Med., 147: 565-568. |
| |
| [32] | Cauthen, G.M., Kilburn, J.O., Kelly, G.D., and Good, R.C. Resistance to anti-tuberculosis drugs in patients with and without prior treatment: survey of 31 state and large city laboratories, 1982-1986. Am. Rev. Respir. Dis., 1988, 137(suppl):260. |
| |
| [33] | Wade, M. M., and Zhang, Y., 2004. Mechanism of drug resistance in Mycobacterium tuberculosis. Frontiers in Bioscience, 9(1), pp.975-994. |
| |
| [34] | Zhang, Y., and Amzel, L M., 2002. Tuberculosis drug targets. Current Drug Targets, 3(2): pp. 131-154. |
| |
| [35] | Zhang, Y., Post-Martens, K., and Denkin, S., 2006. New drug candidates and therapeutic targets for tuberculosis therapy. Drug Discovery Today, 11(1): pp. 21-27. |
| |
| [36] | Tomioka, H., Namba, K., 2006. Development of antitubercular drugs: current status and future prospects, Kekkaku (Japanese Journal)., 81 (12): 753-774. |
| |
| [37] | Zierski, M., and Bek, E., 1980. Side effects of drug regimens used in short-course chemotherapy for pulmonary tuberculosis. Tubercle, 61(1): pp.41-49. |
| |
| [38] | Gray, M.A., 1997. Tuberculosis Drugs. Orthopaedic Nursing, 16(4): 64-69. |
| |
| [39] | Gangadharam, P.R. Isoniazid, rifampin, and hepatotoxicity. Am. Rev. Respir. Dis., 1986, 133:963-965. |
| |
| [40] | Warrington, R.J., Hogg, G.R., Paraskevas, F., and Tse, K.S., 1977. Insidious rifampin-associated renal failure with light-chain proteinuria. Arch. Intern. Med., 137: 927-930. |
| |
| [41] | Zhang, Y., 2005. The magic bullets and tuberculosis drug targets. Annu Rev Pharmacol Toxicol, 45: 529-564. |
| |
| [42] | Garay, S. M. 2004, In Tuberculosis, W. N. a. G. Rom, S.M., ed. (Philadelphia: Lippincott Williams & Wilkins), 345-394. |
| |
| [43] | Gutierrez-Lugo M-T, Bewley CA. Natural Products, Small Molecules, and Genetics in Tuberculosis Drug Development. J. Med. Chem. 51(9), 2606-2612 (2008). |
| |
| [44] | Janin, Y.L. 2007. Antituberculosis drugs: Ten years of research. Bioorg. Med. Chem. 15(7): 2479-2513. |
| |
| [45] | Figueiredo, R., Moiteiro, C., Medeiros, M.A. et al., 2009. Synthesis and evaluation of rifabutin analogs against Mycobacterium avium and H37Rv, MDR and NRP Mycobacterium tuberculosis. Bioorg. Med. Chem. 17(2): 503-511. |
| |
| [46] | Dickinson, J.M., and Mitchison, D. A., 1987. In vitro activity of new rifamycins against rifampicin-resistant M. Tuberculosis and mais-complex Mycobacteria. Tubercle, 68:183-193. |
| |
| [47] | Shoen, C. M., DeStefano, M. S., and Cynamon, M. H.2000. Durable cure for tuberculosis: rifalazil in combination with isoniazid in a murine model of Mycobacterium tuberculosis infection. Clin Infect Dis, 30 Suppl 3, S288-290. |
| |
| [48] | Moghazeh, S. L., Pan, X. S., Arain, T. M., Stover, C. K., and Musser, J. M. Comparative antimycrobial activities of rifampin, rifapentine, and KRM-1648 against a collection of rifampin-resistant Mycobacterium tuberculosis isolates with known rpoB mutations. Antimicrob Agents Chemother, 1996, 40, 2655-2657. |
| |
| [49] | Hidaka, T. 1999. Current status and perspectives on the development of rifamycin derivative antibiotics. Kekkaku, 74 (1): 53-61. |
| |
| [50] | Velayati, A. A., Masjedi, M. R., Farnia, P., Tabarsi, P., Ghanavi, J., Ziazarifi, A. H., and Hoffner, S. E., 2009. Emergence of new forms of totally drug-resistant tuberculosis bacilli: Super extensively drug-resistant tuberculosis or totally drug-resistant strains in Iran. Chest, 136(2): pp.420-425. |
| |
| [51] | Vinšová, J., and Krátký, M., 2010. Tuberculosis - The development of new MDR-TB drugs, In: Drug-Resistant Tuberculosis, Causes, Diagnosis and Treatments, Nguy, S. & K’ung, Z. (Eds.), pp.59-141, Nova Science Publishers, ISBN 978-1-60876-055-8, New York. |
| |
| [52] | Berning, S.E., 2001. The role of fluoroquinolones in tuberculosis today, Drugs. 61: 9-18. |
| |
| [53] | Pasquato KFM, Ferreira EI. An approach for the rational design of new antitubercular agents. Current Drug Targets. 2001, 2: 427-437. |
| |
| [54] | Katz, A. H.; Caufield, C. E. 2003: Structure-based design approaches to cell wall biosynthesis inhibitors. Curr. Pharm. Design. 9: 857-866. |
| |
| [55] | Blanchard, J.S. Molecular mechanisms of drug resistance in Mycobacterium tuberculosis. Annu. Rev. Biochem., 1996, 65:215-239. |
| |
| [56] | Corbett, E. L., Watt, C. J., Walker, N., Maher, D., Williams, B. G., Raviglione, M. C., and Dye, C. 2003. The growing burden of tuberculosis: global trends and interactions with the HIV epidemic. Arch Intern Med, 163, 1009-1021. |
| |
| [57] | Espinal MA. The global situation of MDR-TB. Tuberculosis. 2003, 83: 44-51. |
| |
| [58] | Paramasivan, C. N., Sulochana, S., Kubendiran, G., Venkatesan, P., and Mitchison, D. A. 2005. Bactericidal action of gatifloxacin, rifampin, and isoniazid on logarithmic- and stationary-phase cultures of Mycobacterium tuberculosis. Antimicrob Agents Chemother, 49: 627-631. |
| |
| [59] | Russell, D. G., 2001. Mycobacterium tuberculosis: here today, and here tomorrow. Nat Rev Mol Cell Biol, 2: 569-577. |
| |
| [60] | Smith, C. V., Sharma, V., and Sacchettini, J. C., 2004. TB drug discovery: Addressing issues of persistence and resistance. Tuberculosis, 84, 45-55. |
| |
| [61] | Sunduru, N., Sharma, M., and Chauhan P.M.S., 2010. Recent advances in the design and synthesis of Heterocycles as anti-tubercular agents. Future Med Chem, 2(9): 1469-1500. |
| |